SCHEMBL3884374

SCHEMBL3884374

CNC(=O)c1cc(Oc2ccc3nc(NC[C@H](O)C4CCCCC4)oc3c2)ccn1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 14/20 0.53
BRAF P15056 14/20 0.53
KDR P35968 3/20 0.49
CSF1R P07333 4/20 0.49
PDGFRB P09619 1/20 0.49
KIT P10721 1/20 0.49
PDGFRA P16234 1/20 0.49
FLT3 P36888 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3884227 1.00 RAF1 (0.53) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2677337 0.87 RAF1 (0.66) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2675940 0.87 RAF1 (0.66) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL27759776 0.87 RAF1 (0.51) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2677551 0.87 RAF1 (0.51) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2677540 0.87 RAF1 (0.51) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2675995 0.86 BRAF (0.60) RAF1BRAFKDR
SCHEMBL2678566 0.85 RAF1 (0.54) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2677410 0.85 RAF1 (0.54) RAF1BRAFKDRCSF1RPDGFRB
SCHEMBL2677414 0.85 RAF1 (0.54) RAF1BRAFKDRCSF1RPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010528-A2 6-O-SUBSTITUTED BENZOXAZOLE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF INHIBITING CSF-1R SIGNALING Novartis Pharma AG (CH) 2009-01-07 EP claimed
WO-2007121484-A2 6-O-SUBSTITUTED BENZOXAZOLE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF INHIBITING CSF-1R SIGNALING NOVARTIS AG (CH) 2007-10-25 WO claimed