SCHEMBL3885477

SCHEMBL3885477

CSC(=O)c1[nH]cnc1N

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 1/20 0.60
LMNA P02545 3/20 0.36
KDM4E B2RXH2 3/20 0.36
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PAX8 Q06710 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MMP9 P14780 1/20 0.36
GAA P10253 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 2/20 0.35
KMT2A Q03164 1/20 0.32
XDH P47989 1/20 0.32
MAP3K5 Q99683 1/20 0.32
GABRR1 P24046 1/20 0.31
POLB P06746 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL94902 0.75
SCHEMBL101340 0.75
Hydrochloric Acid SCHEMBL1776088 0.74 GDA (0.96) GDALMNAKDM4ETSHRSMN1; SMN2
SCHEMBL15832982 0.73 GAA (0.39) GDALMNAKDM4ESMN1; SMN2ALDH1A1
SCHEMBL9708864 0.73 GDA (0.60) GDALMNAKDM4ETSHRSMN1; SMN2
SCHEMBL2202786 0.73 GDA (0.60) GDAKDM4ESMN1; SMN2ALDH1A1GAA
SCHEMBL3864458 0.69
SCHEMBL21286900 0.69 GDA (0.60) GDALMNAKDM4ETSHRSMN1; SMN2
Phosphoric Acid SCHEMBL2779124 0.69 GDA (0.85) GDALMNAKDM4ETSHRSMN1; SMN2
SCHEMBL2491314 0.69 KDM4E (0.64) GDALMNAKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140212981-A1 METHODS AND SYSTEMS FOR DETERMINING THE AMOUNT OF THIOPURINE METABOLITES IN A SAMPLE LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2014-07-31 US claimed
WO-2014100405-A1 METHODS AND SYSTEMS FOR DETERMINING THE AMOUNT OF THIOPURINE METABOLITES IN A SAMPLE LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2014-06-26 WO claimed
WO-2016027106-A1 CELL ASSAY UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2016-02-25 WO disclosed
US-20140212981-A1 METHODS AND SYSTEMS FOR DETERMINING THE AMOUNT OF THIOPURINE METABOLITES IN A SAMPLE LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2014-07-31 US disclosed
WO-2014100405-A1 METHODS AND SYSTEMS FOR DETERMINING THE AMOUNT OF THIOPURINE METABOLITES IN A SAMPLE LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2014-06-26 WO disclosed
EP-1825254-A4 METHOD FOR OPTIMIZING THIOPURINE EFFICACY AND TOXICITY USING MASS SPECTROMETRY PROMETHEUS LAB INC (US) 2009-01-14 EP disclosed
EP-1825254-A2 METHOD FOR OPTIMIZING THIOPURINE EFFICACY AND TOXICITY USING MASS SPECTROMETRY Prometheus Laboratories, Inc. (US) 2007-08-29 EP disclosed
US-20060216726-A1 Method for optimizing thiopurine efficacy and toxicity using mass spectrometry PROMETHEUS LABORATORIES INC. (US) 2006-09-28 US disclosed
WO-2006055527-A2 METHOD FOR OPTIMIZING THIOPURINE EFFICACY AND TOXICITY USING MASS SPECTROMETRY PROMETHEUS LABORATORIES INC. (US) 2006-05-26 WO disclosed