SCHEMBL3887929

SCHEMBL3887929

CC(C)c1ccc(-c2cc(N3CCN(c4ncccc4Cl)C[C@H]3C)nc(N3CCOCC3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 9/20 0.48
MTOR P42345 6/20 0.41
PIK3CA P42336 4/20 0.41
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAP3K12 Q12852 1/20 0.38
APAF1 O14727 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3887123 0.93 TRPV1 (0.46) TRPV1MTORPIK3CAMAP3K12
SCHEMBL3889177 0.92 TRPV1 (0.51) TRPV1MTORPIK3CA
SCHEMBL3879587 0.92 TRPV1 (0.42) TRPV1MTORPIK3CAKDM4ELMNA
SCHEMBL3877163 0.91 TRPV1 (0.49) TRPV1MTORPIK3CAKDM4ELMNA
SCHEMBL3876027 0.91 TRPV1 (0.51) TRPV1MTORPIK3CATDP1MAP3K12
SCHEMBL3876090 0.91 TRPV1 (0.47) TRPV1MTORPIK3CAKDM4ELMNA
SCHEMBL13761243 0.90 TRPV1 (0.47) TRPV1MTORPIK3CA
SCHEMBL3879476 0.90 TRPV1 (0.47) TRPV1MTORPIK3CA
SCHEMBL3888987 0.90 TRPV1 (0.47) TRPV1MTORPIK3CA
SCHEMBL3877080 0.90 TRPV1 (0.46) TRPV1MTORPIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed