Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL3903993

CCc1cc([C@@H]2O[C@@H](n3cnc4c(NCC(c5ccccc5)c5ccccc5)nc(N5CCC(NC(=O)Nc6cccnc6)C5)nc43)[C@H](O)C2O)on1.O=C(O)C(F)(F)F

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.46
ADORA3 P0DMS8 4/20 0.42
ADORA1 P30542 4/20 0.42
ADORA2B P29275 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4229411 1.00 ADORA2A (0.46) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2810818 0.97 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL12049816 0.97 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2810816 0.97 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2810819 0.97 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL4130078 0.93 ADORA2A (0.45) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL4130069 0.93 ADORA2A (0.45) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL4130073 0.93 ADORA2A (0.45) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2804820 0.92 ADORA2A (0.50) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2804824 0.92 ADORA2A (0.50) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2018381-A2 USE OF 2-(PURIN-9-YL)-TETRAHYDOFURAN-3,4-DIOL DERIVATIVES AS ADENOSINE A2A RECEPTOR AGONISTS Novartis AG (CH) 2009-01-28 EP disclosed
WO-2007121918-A2 USE OF 2-(PURIN-9-YL)-TETRAHYDOFURAN-3,4-DIOL DERIVATIVES AS ADENOSINE A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2007-11-01 WO disclosed