SCHEMBL3911700

SCHEMBL3911700

CCCCN(Cc1cccc(I)c1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.52
GRIN3B O60391 1/20 0.52
GRIN1 Q05586 1/20 0.52
GRIN2A Q12879 1/20 0.52
GRIN2B Q13224 1/20 0.52
GRIN2C Q14957 1/20 0.52
GRIN3A Q8TCU5 1/20 0.52
PKM P14618 2/20 0.49
HDAC6 Q9UBN7 4/20 0.46
HDAC1 Q13547 3/20 0.46
LTB4R2 Q9NPC1 3/20 0.44
LIMK1 P53667 1/20 0.44
LIMK2 P53671 1/20 0.44
CNR2 P34972 1/20 0.44
HDAC3 O15379 2/20 0.43
HDAC2 Q92769 2/20 0.43
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
LMNA P02545 1/20 0.43
HDAC4 P56524 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17766326 0.90 GRIN2D (0.63) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL1753870 0.85 HDAC6 (0.58) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL27884824 0.83 GRIN2D (0.56) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL27868251 0.79 CYP1A2 (0.60) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7083982 0.79 GRIN2D (0.61) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL15546987 0.79 CNR2 (0.64) PKMHDAC6HDAC1LTB4R2LIMK1
SCHEMBL8773510 0.79 CNR2 (0.64) PKMHDAC6HDAC1LTB4R2LIMK1
SCHEMBL7776491 0.77 CYP1A2 (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7083256 0.77 HDAC1 (0.55) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL25490905 0.76 GRIN2D (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654251-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-03-11 EP disclosed
EP-1654251-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-05-10 EP disclosed
WO-2005016914-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-02-24 WO disclosed