SCHEMBL3913446

SCHEMBL3913446

O=C(NC1CCN(c2ccc(C(=O)O)cn2)CC1)NC1CCN(c2nc(NCC(c3ccccc3)c3ccccc3)c3ncn([C@@H]4O[C@H](COC(=O)C(F)(F)F)[C@H](O)[C@@H]4O)c3n2)C1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.55
NT5E P21589 1/20 0.44
ADORA3 P0DMS8 3/20 0.42
ADORA1 P30542 3/20 0.42
ADORA2B P29275 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4225559 1.00 ADORA2A (0.55) ADORA2ANT5EADORA3ADORA1ADORA2B
Trifluoroacetic Acid SCHEMBL4225568 0.92 ADORA2A (0.62) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL4222343 0.86 ADORA1 (0.53) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL4222703 0.86 ADORA2A (0.51) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL4088376 0.86 ADORA2A (0.51) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL4220361 0.86 ADORA2A (0.51) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL4079238 0.86 ADORA2A (0.51) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL4368669 0.85 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL589286 0.83 ADORA2A (0.43) ADORA2AADORA3ADORA1
Trifluoroacetic Acid SCHEMBL4225494 0.83 ADORA2A (0.73) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2018381-A2 USE OF 2-(PURIN-9-YL)-TETRAHYDOFURAN-3,4-DIOL DERIVATIVES AS ADENOSINE A2A RECEPTOR AGONISTS Novartis AG (CH) 2009-01-28 EP claimed
WO-2007121918-A2 USE OF 2-(PURIN-9-YL)-TETRAHYDOFURAN-3,4-DIOL DERIVATIVES AS ADENOSINE A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2007-11-01 WO claimed