Rivaroxaban

Rivaroxaban

SCHEMBL3914

O=C(NC[C@H]1CN(c2ccc(N3CCOCC3=O)cc2)C(=O)O1)c1ccc(Cl)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

F10

The experimentally established mechanism targets of Rivaroxaban. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F10 known ✓ P00742 20/20 1.00
F2 P00734 2/20 1.00
ABCB11 O95342 1/20 1.00
ST14 Q9Y5Y6 1/20 1.00
CYP1A2 P05177 1/20 0.80
CYP3A4 P08684 1/20 0.80
CYP2D6 P10635 1/20 0.80
CYP2C9 P11712 1/20 0.80
CYP2C19 P33261 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rivaroxaban SCHEMBL77766 1.00 F10 (1.00) F10F2ABCB11ST14CYP1A2
Rivaroxaban SCHEMBL7721848 1.00 F10 (1.00) F10F2ABCB11ST14CYP1A2
Rivaroxaban SCHEMBL14796329 0.99 F10 (0.98) F10F2ABCB11ST14CYP1A2
Rivaroxaban SCHEMBL14796410 0.95 F10 (0.90) F10F2ABCB11ST14CYP1A2
Rivaroxaban SCHEMBL30893049 0.94 F10 (0.90) F10F2ABCB11ST14CYP1A2
SCHEMBL3375861 0.93 F10 (0.86) F10F2ABCB11ST14CYP1A2
SCHEMBL13068882 0.92 F10 (0.85) F10F2ABCB11ST14CYP1A2
SCHEMBL5478295 0.92 F10 (0.85) F10F2ABCB11ST14CYP1A2
Rivaroxaban SCHEMBL12396723 0.91 F10 (0.83) F10F2ABCB11ST14CYP1A2
SCHEMBL20802158 0.91 F10 (0.83) F10F2ABCB11ST14CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 14702 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122084795-A Detection method of rivaroxaban tablet related substances and application thereof 2026-05-26 CN claimed
US-20260137694-A1 NOVEL RIVAROXABAN FORMULATION Shanghai Auson Pharmaceuticals Co., Ltd. (CN) 2026-05-21 US claimed
WO-2026103722-A1 COMPOSITIONS AND METHODS FOR INHIBITING EXPRESSION OF COAGULATION FACTOR XI (FXI) SHANGHAI ARGO BIOPHARMACEUTICAL CO., LTD. (CN) 2026-05-21 WO claimed
CN-119185220-B Rivaroxaban tablet and preparation method thereof 北京悦康科创医药科技股份有限公司 2026-05-15 CN claimed
WO-2026098615-A1 COMPOUND, PHARMACEUTICAL COMPOSITION, AND USE THEREOF IN PREPARATION OF DRUGS FOR TREATING CARDIOVASCULAR AND CEREBROVASCULAR DISEASES 上海东西智荟生物医药有限公司 2026-05-15 WO claimed
EP-4740962-A1 PHARMACEUTICAL COMPOSITION, FORMULATION CONTAINING PHARMACEUTICAL COMPOSITION, KIT CONTAINING PHARMACEUTICAL COMPOSITION, PREPARATION METHOD FOR PHARMACEUTICAL COMPOSITION, AND USE OF PHARMACEUTICAL COMPOSITION Shanghai WD Pharmaceutical Co., Ltd (CN) 2026-05-13 EP claimed
EP-4739305-A1 BUDIODARONE FOR CARDIOVERSION Xyra, LLC (US) 2026-05-13 EP claimed
US-20260124188-A1 mGluR receptor antagonists for use in prevention andor treatment of bone marrow lesions (BML) andor osteoporosis, cartilage loss, osteosclerosis and osteitis in a mammal ORPHELION AB (SE) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4731194-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP Technologies, Inc. (US) 2026-04-29 EP claimed
EP-1685841-A1 Prevention and treatment of thromboembolic disorders Bayer Health Care Aktiengesellschaft (DE) 2006-08-02 EP claimed
WO-2006072367-A1 SOLID, ORALLY APPLICABLE PHARMACEUTICAL ADMINISTRATION FORMS CONTAINING RIVAROXABAN HAVING MODIFIED RELEASE BAYER HEALTHCARE AG (DE) 2006-07-13 WO claimed
WO-2006045756-A1 USE OF DIPYRIDAMOLE IN COMBINATION WITH ANTITHROMBOTICS FOR TREATMENT AND PREVENTION OF THROMBOEMBOLIC DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-05-04 WO claimed
JP-2006513227-A 2006-04-20 JP claimed
EP-1583761-A1 METHOD FOR PRODUCING 5-CHLORO- i N /i -({5 i S /i )-2-OXO-3- 4-(3-OXO-4-MORPHOLINYL)-PHENYL -1,3-OXAZOLIDIN-5-YL&rc ub;-METHYL)-2-THIOPHENE CARBOXAMIDE Bayer HealthCare AG (DE) 2005-10-12 EP claimed
US-20050182055-A1 5-Chloro-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-1,3-oxazolidin-5-yl}methyl)-2-thiophenecarboxamide formed by reacting 4-{4-[(5S)-5-(aminomethyl)-2-oxo-1,3-oxazolidin-3-yl]phenyl}-morpholin-3-one hydrochloride with 5-chlorothiophene-2-carbonyl chloride BAYER HEALTHCARE AG (DE) 2005-08-18 US claimed
WO-2005068456-A1 PRODUCTION METHOD BAYER HEALTHCARE AG (DE) 2005-07-28 WO claimed
US-20050064006-A1 Stents BAYER AKTIENGESELLSCHAFT (DE) 2005-03-24 US claimed
US-20040242660-A1 Combinations of oxazolidinones with other active ingredients for the prophylaxis and/or treatment of thromboembolic disorders BAYER INTELLECTUAL PROPERTY GMBH (DE) 2004-12-02 US claimed
WO-2004060887-A1 METHOD FOR PRODUCING 5-CHLORO-N-({5S)-2-OXO-3-[4-(3-OXO-4-MORPHOLINYL)-PHENYL]-1,3-OXAZOLIDIN-5-YL}-METHYL)-2-THIOPHENE CARBOXAMIDE BAYER HEALTHCARE AG (DE) 2004-07-22 WO claimed