SCHEMBL3917049

SCHEMBL3917049

C[Si](C)(C)CCOC(=O)COc1ccc(N2CC(=O)NS2(=O)=O)c(OCc2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
PTPN2 P17706 1/20 0.35
MET P08581 2/20 0.35
MMP9 P14780 1/20 0.34
ADAM17 P78536 1/20 0.34
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
BCL2 P10415 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3917603 0.86 PTPN1 (0.48) PTPN1KDM4EALDH1A1PTPN2L3MBTL1
SCHEMBL12056117 0.84 PTPN1 (0.41) PTPN1KDM4EALDH1A1MAPTPTPN2
SCHEMBL3917674 0.82 PTPN1 (0.44) PTPN1
SCHEMBL646443 0.77 PTPN1 (0.45) PTPN1ALDH1A1MAPTSMN1; SMN2MMP9
Potassium SCHEMBL646444 0.77 PTPN1 (0.45) PTPN1ALDH1A1MAPTSMN1; SMN2
SCHEMBL4316506 0.77 PTPN1 (0.39) PTPN1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL12056127 0.76 PTPN1 (0.50) PTPN1MAPTPTPN2MAPK1L3MBTL1
SCHEMBL3917446 0.74 PTPN1 (0.47) PTPN1PTPN2
SCHEMBL3920457 0.74 PTPN1 (0.61) PTPN1
SCHEMBL646919 0.74 PTPN1 (0.47) PTPN1ALDH1A1MAPTPTPN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US disclosed
US-20090181928-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-07-16 US disclosed
EP-2038267-A2 THIADIAZOLIDINONE INHIBITORS OF PTPASE Novartis AG (CH) 2009-03-25 EP disclosed
WO-2007115058-A2 THIADIAZOLIDINONE INHIBITORS OF PTPASE NOVARTIS AG (CH) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181928-A1 ORGANIC COMPOUNDS PTPRS, PTPRO, PTPRC PTPN1 21/4885KDM4E 2248/4885LMNA 4825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.