SCHEMBL3919265

SCHEMBL3919265

NC(=O)C[C@H](NC(=O)[C@@H](N)CCC(=O)O)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.51
DPP8 Q6V1X1 2/20 0.51
DPP9 Q86TI2 2/20 0.51
ECE1 P42892 2/20 0.50
GRM8 O00222 1/20 0.50
GRM6 O15303 1/20 0.50
GRIN2D O15399 1/20 0.50
GRIN3B O60391 1/20 0.50
GSR P00390 1/20 0.50
CYP1A2 P05177 1/20 0.50
GRIK1 P39086 1/20 0.50
GRM5 P41594 1/20 0.50
GRIA1 P42261 1/20 0.50
GRIA2 P42262 1/20 0.50
GRIA3 P42263 1/20 0.50
SLC1A3 P43003 1/20 0.50
SLC1A2 P43004 1/20 0.50
SLC1A1 P43005 1/20 0.50
GRIA4 P48058 1/20 0.50
GRIN1 Q05586 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29700608 1.00 DPP4 (0.51) DPP4DPP8DPP9ECE1GRM8
SCHEMBL29517221 1.00 DPP4 (0.51) DPP4DPP8DPP9ECE1GRM8
Hydrochloric Acid SCHEMBL10636183 0.98 DPP4 (0.50) DPP4DPP8DPP9ECE1GRM8
SCHEMBL31339431 0.98 BACE1 (0.51) DPP4DPP8DPP9ECE1GRM8
SCHEMBL29517591 0.95 BACE1 (0.50) DPP4DPP8DPP9ECE1GRM8
SCHEMBL31314398 0.95 BACE1 (0.49) DPP4DPP8DPP9ECE1GRM8
SCHEMBL30423552 0.95 BACE1 (0.49) DPP4DPP8DPP9ECE1GRM8
SCHEMBL29575299 0.95 BACE1 (0.50) DPP4DPP8DPP9ECE1GRM8
SCHEMBL30596289 0.93 BACE1 (0.48) DPP4DPP8DPP9ECE1GRM8
SCHEMBL30553776 0.92 BACE1 (0.50) DPP4DPP8DPP9ECE1GRM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4036149-B1 HETEROBIFUNCTIONAL MONODISPERSED POLYETHYLENE GLYCOL HAVING PEPTIDE LINKER NOF CORP (JP) 2026-04-29 EP claimed
WO-2025245258-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONIST ANALOGS FOR MODULATING WEIGHT GAIN ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245279-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USE THEREFORE IN TREATMENT OF ADDICTION AND/OR PAIN ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245294-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USES THEREOF FOR MODULATING WEIGHT GAIN ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245244-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONIST ANALOGS FOR MODULATING WEIGHT LOSS ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245292-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USES THEREOF FOR MODULATING WEIGHT LOSS ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
WO-2025245252-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONIST ANALOGS FOR USE IN PAIN MANAGEMENT AND/OR SUBSTANCE USE DISORDERS ENDEVICA BIO, INC. (US) 2025-11-27 WO claimed
EP-3649146-B1 APELIN PEPTIDES AND USES THEREOF UNIV ALBERTA (CA) 2024-06-26 EP claimed
EP-3938372-B1 AZETIDOBENZODIAZEPINE DIMERS AND CONJUGATES COMPRISING THEM FOR USE IN THE TREATMENT OF CANCER MEDIMMUNE LTD (GB) 2023-10-25 EP claimed
US-11753445-B2 Therapeutic peptides COHBAR, INC. (US) 2023-09-12 US claimed
CN-116410961-A Tobacco etching virus protease fusion protein and preparation method and application thereof 重庆艾力彼生物科技有限公司 2023-07-11 CN claimed
US-20220242912-A1 THERAPEUTIC PEPTIDES COHBAR, INC. 2022-08-04 US claimed
US-11332497-B2 Therapeutic peptides COHBAR, INC. (US) 2022-05-17 US claimed
EP-3546448-B1 DI-SUBSTITUTED MALEIC AMIDE LINKER FOR ANTIBODY-DRUG CONJUGATING AND PREPARATION METHOD AND USE THEREOF MABWELL SHANGHAI BIOSCIENCE CO LTD (CN) 2022-04-06 EP claimed
EP-4684030-A2 METHOD OF DEPROTECTING AT LEAST ONE D-AMINO ACID AND/OR D-AMINO ACID DERIVATIVE PROTECTED FUNCTIONAL GROUP Martin-Luther-Universität Halle-Wittenberg (DE) 2026-01-28 EP disclosed
WO-2025245244-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONIST ANALOGS FOR MODULATING WEIGHT LOSS ENDEVICA BIO, INC. (US) 2025-11-27 WO disclosed
WO-2025245294-A1 NON-NATURALLY OCCURRING MELANOCORTIN RECEPTOR AGONISTS AND USES THEREOF FOR MODULATING WEIGHT GAIN ENDEVICA BIO, INC. (US) 2025-11-27 WO disclosed
US-4731412-A Process and composition for amino-terminal, α-aspartyl and α-glutamyl dipeptide esters THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1988-03-15 US disclosed
US-4600532-A Process and composition for amino-terminal, α-aspartyl and α-glutamyl dipeptides and dipeptide esters THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1986-07-15 US disclosed
US-4600532-A Process and composition for amino-terminal, α-aspartyl and α-glutamyl dipeptides and dipeptide esters THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1986-07-15 US disclosed