SCHEMBL3922080

SCHEMBL3922080

COc1ccc(-c2ccc3nc(N)nc(N4CCC(NC(=O)OC(C)(C)C)C4)c3n2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
CFTR P13569 3/20 0.47
AURKA O14965 3/20 0.47
PDPK1 O15530 3/20 0.47
AURKB Q96GD4 3/20 0.47
SUV39H2 Q9H5I1 10/20 0.45
MAP4K4 O95819 2/20 0.44
NOS1 P29475 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4121554 1.00 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DCFTR
SCHEMBL3921361 1.00 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DCFTR
SCHEMBL3924839 0.87 MAP4K4 (0.47) PDE4APDE4BPDE4CPDE4DAURKA
SCHEMBL3927951 0.87 MAP4K4 (0.47) PDE4APDE4BPDE4CPDE4DAURKA
SCHEMBL3929667 0.82 MAP4K4 (0.51) AURKAPDPK1AURKBSUV39H2MAP4K4
SCHEMBL8153360 0.82 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DNOS1
SCHEMBL8152356 0.82 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DNOS1
SCHEMBL4001268 0.81 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DNOS1
SCHEMBL8256368 0.81 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DNOS1
SCHEMBL3931773 0.81 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DSUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009003669-A2 PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR MEDICAL TREATMENT 4 AZA IP NV (BE) 2009-01-08 WO disclosed