SCHEMBL3924880

SCHEMBL3924880

CC(C)(C)OC(=O)N1CCC(COCCc2cc(Cl)cc3cn[nH]c23)(c2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACACB O00763 7/20 0.46
TACR1 P25103 4/20 0.42
NAMPT P43490 2/20 0.38
SLC6A4 P31645 3/20 0.38
KCNH2 Q12809 3/20 0.38
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
IDO1 P14902 1/20 0.35
CCR5 P51681 2/20 0.35
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2423912 0.84 ACACB (0.45) ACACBTACR1NAMPTHDAC1HDAC2
SCHEMBL2430727 0.83 ACACB (0.44) ACACBTACR1NAMPTHDAC1HDAC2
SCHEMBL2424824 0.83 ACACB (0.44) ACACBTACR1NAMPTHDAC1HDAC2
SCHEMBL2424822 0.83 ACACB (0.44) ACACBTACR1NAMPTHDAC1HDAC2
SCHEMBL2425177 0.82 TACR1 (0.57) ACACBTACR1SLC6A4KCNH2
SCHEMBL2424827 0.82 ACACB (0.43) ACACBTACR1NAMPTSLC6A4KCNH2
SCHEMBL3932000 0.82 TACR1 (0.38) ACACBTACR1SLC6A4KCNH2
SCHEMBL2424361 0.81 ACACB (0.43) ACACBTACR1NAMPTHDAC1HDAC2
SCHEMBL2424900 0.81 ACACB (0.43) ACACBTACR1NAMPTHDAC1HDAC2
SCHEMBL2430951 0.81 ACACB (0.43) ACACBTACR1NAMPTHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed