SCHEMBL3925967

SCHEMBL3925967

C[Si](C)(C)CCOCn1nc2c(CCOCC3(c4ccccc4)CCN(C(=O)O)CC3)cc(C(F)(F)F)cc2c1C#N

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.43
SLC6A4 P31645 3/20 0.40
KCNH2 Q12809 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3925072 0.91 TACR1 (0.46) TACR1SLC6A4KCNH2
SCHEMBL3935350 0.90 TACR1 (0.45) TACR1SLC6A4KCNH2
SCHEMBL2425049 0.86 TACR1 (0.40) TACR1SLC6A4KCNH2
SCHEMBL2430916 0.84 TACR1 (0.50) TACR1SLC6A4KCNH2
SCHEMBL2430705 0.84 TACR1 (0.49) TACR1SLC6A4KCNH2
SCHEMBL3936516 0.83 TACR1 (0.46) TACR1SLC6A4KCNH2
SCHEMBL4005593 0.82 TACR1 (0.47) TACR1SLC6A4KCNH2
SCHEMBL2430877 0.81 TACR1 (0.47) TACR1SLC6A4KCNH2
SCHEMBL3925517 0.80 TACR1 (0.40) TACR1SLC6A4KCNH2
SCHEMBL12290307 0.78 TACR1 (0.59) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed