SCHEMBL3926055

SCHEMBL3926055

COc1cc(CCOCC2(c3ccc(F)cc3)CCN(C(=O)O)CC2)c2nn(COCC[Si](C)(C)C)cc2c1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.35
SLC6A4 P31645 17/20 0.35
KCNH2 Q12809 17/20 0.35
NQO2 P16083 1/20 0.34
PTGER2 P43116 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
LTB4R Q15722 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
S1PR1 P21453 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3934661 0.93 TACR1 (0.35) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3925634 0.91 TACR1 (0.34) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3937267 0.90 TACR1 (0.34) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3938855 0.90 TACR1 (0.36) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3934408 0.89 TACR1 (0.33) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3926165 0.89 TACR1 (0.42) TACR1SLC6A4KCNH2
SCHEMBL3925731 0.88 TACR1 (0.43) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3926288 0.88 TACR1 (0.41) TACR1SLC6A4KCNH2S1PR1
SCHEMBL3935292 0.87 TACR1 (0.33) TACR1SLC6A4KCNH2S1PR1
SCHEMBL2433923 0.85 TACR1 (0.33) TACR1SLC6A4KCNH2NQO2PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed