SCHEMBL3926070

SCHEMBL3926070

CC(C)(C)OC(=O)N1CCC(COCCc2cc(Cl)cc3c(Br)n(COCC[Si](C)(C)C)nc23)(c2ccc(F)cc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.38
HDAC2 Q92769 2/20 0.34
HDAC1 Q13547 1/20 0.34
PARP1 P09874 3/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
TNKS O95271 2/20 0.32
TNKS2 Q9H2K2 2/20 0.32
PKM P14618 1/20 0.32
JAK2 O60674 2/20 0.32
JAK1 P23458 2/20 0.32
NAMPT P43490 1/20 0.32
TP53 P04637 1/20 0.31
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3927297 0.93 TACR1 (0.40) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL3931010 0.89 TACR1 (0.35) TACR1SLC6A4KCNH2
SCHEMBL2429952 0.87 TACR1 (0.35) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL2429954 0.87 TACR1 (0.35) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL3937761 0.82 TACR1 (0.38) TACR1HDAC2HDAC1CNR1CNR2
SCHEMBL2425718 0.80 TACR1 (0.37) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL2425716 0.80 TACR1 (0.37) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL2426430 0.79 TACR1 (0.35) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL2428513 0.79 TACR1 (0.35) TACR1HDAC2HDAC1PARP1CNR1
SCHEMBL12290304 0.79 TACR1 (0.58) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed