SCHEMBL3928951

SCHEMBL3928951

CC(C)(C)OC(=O)N1CCC(COCC(C#N)c2cc(Cl)cc3cn(COCC[Si](C)(C)C)nc23)(c2ccc(F)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.36
JAK2 O60674 11/20 0.36
JAK1 P23458 11/20 0.36
SLC6A4 P31645 2/20 0.34
KCNH2 Q12809 2/20 0.34
F2RL1 P55085 1/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3923286 0.91 TACR1 (0.38) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL3934412 0.91 TACR1 (0.38) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL2425983 0.90 JAK2 (0.38) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL3926859 0.90 TACR1 (0.37) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL2423310 0.88 JAK2 (0.36) TACR1JAK2JAK1
SCHEMBL3935599 0.88 TACR1 (0.37) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL12290807 0.88 TACR1 (0.37) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL12290455 0.88 TACR1 (0.37) TACR1JAK2JAK1SLC6A4KCNH2
SCHEMBL3923863 0.87 TACR1 (0.35) TACR1SLC6A4KCNH2F2RL1CNR1
SCHEMBL2427186 0.87 TACR1 (0.37) TACR1JAK2JAK1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed