SCHEMBL3929924

SCHEMBL3929924

N#Cc1ccc(N2CC(=O)NS2(=O)=O)c(OCc2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.45
MAOB P27338 1/20 0.41
SLC6A9 P48067 1/20 0.39
PTGER1 P34995 1/20 0.38
HTR6 P50406 2/20 0.38
MRGPRX4 Q96LA9 4/20 0.38
TDP2 O95551 3/20 0.37
KCNH2 Q12809 1/20 0.37
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
HTR1A P08908 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
EGLN2 Q96KS0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920457 0.84 PTPN1 (0.61) PTPN1MRGPRX4HTR1ASLC6A2SLC6A4
SCHEMBL3917425 0.84 PTPN1 (0.47) PTPN1PTGER1MRGPRX4SLC6A4
SCHEMBL12056127 0.84 PTPN1 (0.50) PTPN1MAOBPTGER1HTR6MRGPRX4
SCHEMBL646919 0.84 PTPN1 (0.47) PTPN1HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL3917446 0.84 PTPN1 (0.47) PTPN1HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL3926449 0.83 PTPN1 (0.43) PTPN1MAOB
SCHEMBL3917216 0.83 PTPN1 (0.41) PTPN1MAOB
SCHEMBL647271 0.82 PTPN1 (0.44) PTPN1MRGPRX4PDCD1CD274
SCHEMBL4443447 0.82 PTPN1 (0.46) PTPN1
SCHEMBL3917279 0.82 PTPN1 (0.46) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US disclosed
US-20090181928-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-07-16 US disclosed
EP-2038267-A2 THIADIAZOLIDINONE INHIBITORS OF PTPASE Novartis AG (CH) 2009-03-25 EP disclosed
WO-2007115058-A2 THIADIAZOLIDINONE INHIBITORS OF PTPASE NOVARTIS AG (CH) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181928-A1 ORGANIC COMPOUNDS PTPRS, PTPRO, PTPRC PTPN1 21/4885MAOB 1270/4885SLC6A9 4588/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.