SCHEMBL3933743

SCHEMBL3933743

CCOC(=Nc1cc(Cl)cc2cn(C3CC3)nc12)C(Cl)(Cl)Cl

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 6/20 0.33
TLR7 Q9NYK1 4/20 0.32
TLR9 Q9NR96 3/20 0.32
TLR4 O00206 2/20 0.32
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13961185 0.66 TLR8 (0.36) TLR8TLR7TLR9TLR4DRD2
SCHEMBL2428960 0.66 GRM2 (0.38) TLR8TLR7TLR9TLR4DRD2
SCHEMBL24447954 0.59 PDE4D (0.36) TLR8TLR7TLR9TLR4IRAK4
SCHEMBL1407155 0.59 BAZ2B (0.43)
SCHEMBL25341920 0.59 MAPT (0.39) IRAK4
SCHEMBL25113904 0.58 PDE4D (0.43) TLR8TLR7TLR9TLR4IRAK4
SCHEMBL26762008 0.57 TLR8 (0.42) TLR8TLR7TLR9TLR4
SCHEMBL26352388 0.56 PDE4D (0.39) TLR8TLR7TLR9TLR4
SCHEMBL1407057 0.56 BAZ2B (0.39)
SCHEMBL24345435 0.56 PDE4D (0.43) TLR8TLR7TLR9TLR4IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed