SCHEMBL3936713

SCHEMBL3936713

CCCCC#Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.45
FFAR1 O14842 1/20 0.44
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
PTPN1 P18031 1/20 0.41
KCNH2 Q12809 2/20 0.40
PTGES O14684 1/20 0.39
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
ADORA2B P29275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3937119 0.90 GRM5 (0.47) GRM5FFAR1PTPN1PTGESALDH1A1
SCHEMBL2951986 0.84 FFAR1 (0.47) GRM5FFAR1PTPN1KCNH2PTGES
SCHEMBL4174001 0.83 GRM5 (0.49) GRM5FFAR1PTPN1PTGES
SCHEMBL2946792 0.83 HTR2C (0.48) GRM5FFAR1PTPN1KCNH2PTGES
SCHEMBL5092655 0.81 GRM5 (0.40) GRM5FFAR1HDAC3HDAC1HDAC2
SCHEMBL5092664 0.81 GRM5 (0.40) GRM5FFAR1HDAC3HDAC1HDAC2
SCHEMBL2950490 0.81 FFAR1 (0.49) GRM5FFAR1PTPN1PTGES
SCHEMBL2236377 0.81 FFAR1 (0.53) GRM5FFAR1HDAC1PTPN1PTGES
SCHEMBL3940735 0.80 FFAR1 (0.43) FFAR1KCNH2
SCHEMBL7517707 0.80 FFAR1 (0.62) FFAR1PTPN1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046746-A2 CHEMICAL COMPOUNDS Praecis Pharmaceuticals Incorporated (US) 2009-04-15 EP disclosed
WO-2008016692-A2 CHEMICAL COMPOUNDS PRAECIS PHARMACEUTICALS INCORPORATED (US) 2008-02-07 WO disclosed