SCHEMBL3942284

SCHEMBL3942284

COc1cncc(NC(=O)c2cc(NC(=O)c3cccc(C(C)(C)C#N)c3F)ccc2C)c1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRAF P15056 19/20 0.71
CYP2C9 P11712 5/20 0.56
LCK P06239 1/20 0.44
BTK Q06187 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3940175 0.85 BRAF (0.69) BRAFCYP2C9
SCHEMBL3939889 0.83 BRAF (1.00) BRAFCYP2C9LCKBTK
SCHEMBL3938207 0.75 BRAF (0.72) BRAFCYP2C9LCKBTK
SCHEMBL3934779 0.75 BRAF (0.77) BRAFCYP2C9LCKBTK
SCHEMBL4167730 0.75 BRAF (0.84) BRAFCYP2C9LCK
SCHEMBL4788091 0.74 BRAF (0.51) BRAF
SCHEMBL3934034 0.74 BRAF (0.83) BRAFCYP2C9LCKBTK
SCHEMBL4175332 0.74 BRAF (0.67) BRAFCYP2C9LCKBTK
SCHEMBL3934373 0.74 BRAF (0.71) BRAFCYP2C9LCKBTK
SCHEMBL3934259 0.74 BRAF (0.82) BRAFCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed