SCHEMBL3949080

SCHEMBL3949080

N=c1[nH]cccc1F

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27851304 0.69 JAK2 (0.39)
SCHEMBL16445619 0.69 KDM4E (0.39)
SCHEMBL8091109 0.68
SCHEMBL30475376 0.68
SCHEMBL4240507 0.68
SCHEMBL482079 0.68
SCHEMBL2662014 0.68
SCHEMBL17037403 0.68
Iodide SCHEMBL11482211 0.67
SCHEMBL1894921 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080145514-A1 Compositions and methods for coating medical implants ANGIOTECH INTERNATIONAL AG (CH) 2008-06-19 US claimed
US-20080113000-A1 Compositions and methods for coating medical implants ANGIOTECH INTERNATIONAL AG (CH) 2008-05-15 US claimed
EP-3204043-B1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF CANCER WITH 5-IODO-2-PYRIMIDINONE-2'-DEOXYRIBOSE (IPdR) KINSELLA TIMOTHY J (US) 2023-06-07 EP disclosed
EP-3204043-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF CANCER WITH 5-IODO-2-PYRIMIDINONE-2'-DEOXYRIBOSE (IPdR) Kinsella, Timothy J. (US) 2017-08-16 EP disclosed
WO-2016057699-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF CANCER WITH 5-IODO-2-PYRIMIDINONE-2'-DEOXYRIBOSE (IPdR) KINSELLA TIMOTHY J (US) 2016-04-14 WO disclosed
EP-1774039-A4 GENETIC MARKERS FOR PREDICTING DISEASE AND TREATMENT OUTCOME UNIV SOUTHERN CALIFORNIA (US) 2009-07-08 EP disclosed
EP-1774039-A2 GENETIC MARKERS FOR PREDICTING DISEASE AND TREATMENT OUTCOME UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2007-04-18 EP disclosed
US-20060115827-A1 Genetic markers for predicting disease and treatment outcome UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2006-06-01 US disclosed
WO-2006012361-A2 GENETIC MARKERS FOR PREDICTING DISEASE AND TREATMENT OUTCOME UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2006-02-02 WO disclosed