SCHEMBL3949196

SCHEMBL3949196

COC[C@H]1C[C@H](O[Si](C)(C)C(C)(C)C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.35
ABCB1 P08183 1/20 0.34
UCHL1 P09936 1/20 0.33
PDE4B Q07343 1/20 0.33
PARP1 P09874 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SRC P12931 8/20 0.31
CYP1A2 P05177 1/20 0.30
POLB P06746 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30
GPR119 Q8TDV5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24894673 1.00 NR1H2 (0.35) NR1H2ABCB1UCHL1PDE4BPARP1
SCHEMBL2387181 1.00 NR1H2 (0.35) NR1H2ABCB1UCHL1PDE4BPARP1
SCHEMBL9383410 1.00 NR1H2 (0.35) NR1H2ABCB1UCHL1PDE4BPARP1
SCHEMBL24826386 1.00 NR1H2 (0.35) NR1H2ABCB1UCHL1PDE4BPARP1
SCHEMBL12553792 1.00 NR1H2 (0.35) NR1H2ABCB1UCHL1PDE4BPARP1
SCHEMBL8759166 0.91 NR1H2 (0.32) NR1H2ABCB1PARP1
SCHEMBL8759141 0.91 NR1H2 (0.32) NR1H2ABCB1PARP1
SCHEMBL12519787 0.90 NR1H2 (0.33) NR1H2ABCB1UCHL1PARP1CHRM2
SCHEMBL1526484 0.90 NR1H2 (0.35) NR1H2ABCB1PARP1CHRM2CHRM1
SCHEMBL1526483 0.90 NR1H2 (0.35) NR1H2ABCB1PARP1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026197-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE GLAXO GROUP LIMITED (GB) 2009-02-26 WO disclosed