SCHEMBL3961277

SCHEMBL3961277

CCN(CC)CCOc1cc(-c2nc(SCC(=O)N(C)C)nc3[nH]cc(C#N)c23)c(Cl)cc1OC

nearest known ligand 0.83

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.83
HSP90AB1 P08238 15/20 0.73
KCNH2 Q12809 5/20 0.73
SMN1; SMN2 Q16637 1/20 0.36
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3950788 0.91 HSP90AA1 (1.00) HSP90AA1HSP90AB1KCNH2SMN1; SMN2
SCHEMBL3956794 0.85 HSP90AA1 (0.89) HSP90AA1HSP90AB1KCNH2SMN1; SMN2
SCHEMBL2563125 0.85 HSP90AB1 (0.72) HSP90AA1HSP90AB1KCNH2
SCHEMBL2562465 0.84 HSP90AB1 (1.00) HSP90AA1HSP90AB1KCNH2CYP2C19
SCHEMBL2565891 0.84 HSP90AB1 (1.00) HSP90AA1HSP90AB1KCNH2
SCHEMBL12161130 0.83 HSP90AB1 (0.74) HSP90AA1HSP90AB1KCNH2
SCHEMBL12161039 0.82 HSP90AB1 (0.69) HSP90AA1HSP90AB1KCNH2
SCHEMBL3961384 0.82 HSP90AB1 (0.92) HSP90AA1HSP90AB1KCNH2
SCHEMBL3950781 0.81 HSP90AB1 (0.74) HSP90AA1HSP90AB1KCNH2
SCHEMBL3958501 0.81 HSP90AB1 (0.74) HSP90AA1HSP90AB1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO claimed
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO disclosed
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO disclosed