SCHEMBL3973176

SCHEMBL3973176

Cc1ccc(NC(=O)c2ccnc(Cl)c2)cc1Nc1nccc(-c2cccnc2)n1

nearest known ligand 0.82

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 13/20 0.82
PDGFRA P16234 11/20 0.82
BCR P11274 7/20 0.82
PDGFRB P09619 5/20 0.82
EGFR P00533 1/20 0.80
PRKCA P17252 1/20 0.80
KIT P10721 7/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3219611 0.90 PDGFRA (0.83) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL9677 0.90 PDGFRA (1.00) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL2004455 0.90 PDGFRA (0.91) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL13492414 0.89 ABL1 (0.80) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL9782 0.89 PDGFRA (1.00) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL29498750 0.89 PDGFRA (1.00) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL11932096 0.88 PDGFRA (0.86) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL4802851 0.88 ABL1 (0.83) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL1656154 0.88 PDGFRA (0.90) ABL1PDGFRABCRPDGFRBEGFR
SCHEMBL13492339 0.88 ABL1 (0.74) ABL1PDGFRABCRPDGFRBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100048539-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2010-02-25 US disclosed
US-20100048539-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2010-02-25 US disclosed
EP-2079729-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-07-22 EP disclosed
WO-2008058037-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-05-15 WO disclosed
WO-2008058037-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048539-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS PDGFRB, PDGFRA, KIT ABL1 9/4885PDGFRA 2/4885BCR 65/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.