SCHEMBL3975154

SCHEMBL3975154

CCN1C(=O)N(c2cc(OC)cc(OC)c2C)Cc2cnc(Nc3ccncc3)nc21

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 13/20 0.49
TNK2 Q07912 1/20 0.44
MAP4K2 Q12851 1/20 0.44
FGFR1 P11362 5/20 0.43
FGFR2 P21802 4/20 0.43
FGFR3 P22607 4/20 0.43
BMX P51813 3/20 0.41
EGFR P00533 3/20 0.41
CSF1R P07333 2/20 0.41
FYN P06241 1/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
MAPK1 P28482 1/20 0.40
KDR P35968 1/20 0.40
EPHB3 P54753 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3968638 0.91 FGFR4 (0.53) FGFR4TNK2MAP4K2FGFR1FGFR2
SCHEMBL3976274 0.88 FGFR4 (0.48) FGFR4TNK2MAP4K2FGFR1FGFR2
SCHEMBL3968277 0.87 FGFR4 (0.65) FGFR4TNK2MAP4K2FGFR1FGFR2
SCHEMBL3977362 0.86 LCK (0.55) FGFR4TNK2MAP4K2FGFR1FGFR2
SCHEMBL3970490 0.85 FGFR1 (0.45) FGFR4FGFR1FGFR2FGFR3
SCHEMBL3968636 0.82 EGFR (0.53) FGFR4FGFR1FGFR2FGFR3EGFR
SCHEMBL3970204 0.82 FGFR4 (0.59) FGFR4FGFR1FGFR2FGFR3
SCHEMBL3972202 0.79 FGFR4 (0.51) FGFR4TNK2MAP4K2FGFR1FGFR2
SCHEMBL3972965 0.78 LCK (0.58) FGFR4TNK2MAP4K2FGFR1FGFR2
SCHEMBL3975643 0.76 FGFR1 (0.49) FGFR4FGFR1FGFR2FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7501425-B1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyprimidines as inhibitors of cellular proliferation WARNER LAMBERT COMPANY (US) 2009-03-10 US claimed
EP-1801112-A1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation Warner-Lambert Company LLC (US) 2007-06-27 EP claimed
US-7501425-B1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyprimidines as inhibitors of cellular proliferation WARNER LAMBERT COMPANY (US) 2009-03-10 US disclosed
EP-1801112-A1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation Warner-Lambert Company LLC (US) 2007-06-27 EP disclosed
US-20040044012-A1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation DOBRUSIN ELLEN MYRA (US) 2004-03-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040044012-A1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation CCNI, CCNH, CCNA1 FGFR4 95/4885TNK2 277/4885MAP4K2 586/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.