SCHEMBL3977699

SCHEMBL3977699

O=C(O)NC1CC2CCC(C1)N2c1ccc(C(=O)NCc2ccccc2)cn1

nearest known ligand 0.80

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 12/20 0.80
HSP90AB1 P08238 12/20 0.80
ALDH1A1 P00352 2/20 0.55
RAB9A P51151 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MAPK1 P28482 2/20 0.55
KDM4E B2RXH2 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.53
HPGDS O60760 3/20 0.49
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3977695 1.00 HSP90AA1 (0.80) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2429288 0.89 HSP90AA1 (1.00) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2429285 0.89 HSP90AA1 (1.00) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2429123 0.89 HSP90AA1 (1.00) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2429124 0.89 HSP90AA1 (1.00) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2427601 0.88 HSP90AA1 (0.88) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2427598 0.88 HSP90AA1 (0.88) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2430973 0.87 HSP90AA1 (0.74) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2430971 0.87 HSP90AA1 (0.74) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL2424281 0.87 HSP90AA1 (0.82) HSP90AA1HSP90AB1ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed