SCHEMBL3978463

SCHEMBL3978463

Cc1cc(C(O)(C(F)(F)F)C(F)(F)F)ccc1OCc1nc(-c2cccc(Cl)c2)oc1C

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.61
NR1H3 Q13133 6/20 0.61
PPARG P37231 3/20 0.43
PPARA Q07869 3/20 0.43
CYP2C9 P11712 1/20 0.43
KCNH2 Q12809 1/20 0.43
KDR P35968 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
PPARD Q03181 1/20 0.41
MAPT P10636 3/20 0.41
TP53 P04637 2/20 0.41
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980129 0.93 NR1H2 (0.65) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3976062 0.90 NR1H2 (0.50) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3984282 0.89 NR1H2 (0.61) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3976394 0.88 NR1H2 (0.66) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3979271 0.87 NR1H2 (0.60) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3977183 0.86 NR1H2 (0.45) NR1H2NR1H3PPARGPPARAPPARD
SCHEMBL3979351 0.86 NR1H2 (0.56) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3978464 0.85 NR1H2 (0.66) NR1H2NR1H3PPARGPPARAMAPK1
SCHEMBL3981231 0.83 NR1H2 (0.45) NR1H2NR1H3PPARGPPARACYP2C9
SCHEMBL3977264 0.83 NR1H2 (0.53) NR1H2NR1H3KDRMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101031540-B Hexafluoroisopropanol substituted ether derivatives HOFFMANN LA ROCHE 2010-05-26 CN claimed
US-7473705-B2 Hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. (US) 2009-01-06 US claimed
EP-1802566-B1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-11-26 EP claimed
CN-101031540-A Hexafluoroisopropanol substituted ether derivatives HOFFMANN LA ROCHE (CH) 2007-09-05 CN claimed
EP-1802566-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-07-04 EP claimed
WO-2006037480-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-04-13 WO claimed
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. 2006-04-06 US claimed
CN-101031540-B Hexafluoroisopropanol substituted ether derivatives HOFFMANN LA ROCHE 2010-05-26 CN disclosed
US-7473705-B2 Hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. (US) 2009-01-06 US disclosed
EP-1802566-B1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-11-26 EP disclosed
CN-101031540-A Hexafluoroisopropanol substituted ether derivatives HOFFMANN LA ROCHE (CH) 2007-09-05 CN disclosed
EP-1802566-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-07-04 EP disclosed
WO-2006037480-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-04-13 WO disclosed
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. 2006-04-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives NR1H3, NR1H2, NR1I2 NR1H2 2/4885NR1H3 1/4885PPARG 22/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.