SCHEMBL3979751

SCHEMBL3979751

FC(F)(F)c1ccc([C@@]23C[C@H]2CN(CCCSc2ncccn2)C3)cc1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.68
KCNH2 Q12809 20/20 0.68
DRD2 P14416 15/20 0.68
CYP1A2 P05177 1/20 0.60
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3555210 1.00 DRD3 (0.68) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL3979750 1.00 DRD3 (0.68) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL3545896 0.88 DRD3 (0.63) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL13312911 0.88 DRD3 (0.57) DRD3KCNH2DRD2CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL3550781 0.88 DRD3 (0.62) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL2822280 0.85 DRD3 (0.61) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL2818581 0.84 DRD3 (0.66) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL2819170 0.84 DRD3 (0.62) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL2822383 0.84 DRD3 (0.59) DRD3KCNH2DRD2CYP1A2CYP2C19
SCHEMBL13312910 0.83 DRD3 (0.58) DRD3KCNH2DRD2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926723-B1 AZABICYCLO (3,1,0) HEXAN DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RCEPTORS GLAXO GROUP LTD (GB) 2009-05-13 EP claimed