SCHEMBL3986388

SCHEMBL3986388

CCc1cc(Cc2ccc(F)c(C(=O)N3CCC4(CCCN4)CC3)c2)n[nH]c1=O

nearest known ligand 0.72

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.72
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4248742 0.95 PARP1 (0.66) PARP1KCNH2
SCHEMBL20544239 0.86 PARP1 (0.65) PARP1
SCHEMBL20544682 0.85 PARP1 (0.73) PARP1
SCHEMBL20544688 0.84 PARP1 (0.68) PARP1
SCHEMBL20544503 0.84 PARP1 (1.00) PARP1
SCHEMBL3920570 0.83 PARP1 (0.68) PARP1
Trifluoroacetic Acid SCHEMBL3916008 0.81 PARP1 (0.59) PARP1
Trifluoroacetic Acid SCHEMBL3980202 0.81 PARP1 (0.67) PARP1
Trifluoroacetic Acid SCHEMBL3085468 0.80 PARP1 (0.62) PARP1
SCHEMBL20544245 0.80 PARP1 (1.00) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029551-B1 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) MSD ITALIA SRL (IT) 2018-10-31 EP claimed
EP-2029551-A2 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2009-03-04 EP disclosed
WO-2007138351-A2 PYRIDINONE AND PYRIDAZINONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-12-06 WO disclosed