SCHEMBL4010890

SCHEMBL4010890

O=C(O)CCCCOc1ncc(C(=O)NC2CCCC[C@H]2O)cc1-c1ccc(Cl)cc1

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 0.82
TACR2 P21452 1/20 0.80
CNR2 P34972 2/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2704550 1.00 CNR1 (0.82) CNR1TACR2CNR2
SCHEMBL1378063 0.93 CNR1 (0.82) CNR1TACR2CNR2
SCHEMBL1378062 0.93 CNR1 (0.82) CNR1TACR2CNR2
SCHEMBL2705566 0.91 CNR1 (0.84) CNR1TACR2CNR2
SCHEMBL2704102 0.90 CNR1 (1.00) CNR1TACR2CNR2
SCHEMBL1377904 0.90 CNR1 (0.91) CNR1TACR2CNR2
SCHEMBL1377255 0.89 CNR1 (1.00) CNR1TACR2CNR2
SCHEMBL5271693 0.89 CNR1 (1.00) CNR1TACR2CNR2
SCHEMBL1377250 0.89 CNR1 (1.00) CNR1TACR2CNR2
SCHEMBL1376708 0.89 CNR1 (1.00) CNR1TACR2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074096-A1 3-PYRIDINECARBOXAMIDE AND 2-PYRAZINECARBOXAMIDE DERIVATIVES AS HDL-CHOLESTEROL RAISING AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2009-07-01 EP disclosed
WO-2008040651-A1 3-PYRIDINECARBOXAMIDE AND 2-PYRAZINECARBOXAMIDE DERIVATIVES AS HDL-CHOLESTEROL RAISING AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-04-10 WO disclosed