SCHEMBL4013665

SCHEMBL4013665

CCS(=O)(=O)c1cc(-c2cccc(-c3ccnc4c(C(F)(F)F)cccc34)c2)ccc1C

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 19/20 0.74
NR1H3 Q13133 16/20 0.74
RXRA P19793 1/20 0.53
PPARG P37231 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013215 0.89 NR1H2 (0.80) NR1H2NR1H3RXRA
SCHEMBL4011381 0.89 NR1H2 (0.72) NR1H2NR1H3RXRAPPARG
SCHEMBL4010780 0.88 NR1H2 (0.61) NR1H2NR1H3RXRAPPARGPTGDR2
SCHEMBL4011921 0.87 NR1H2 (0.72) NR1H2NR1H3RXRAPPARG
SCHEMBL4010294 0.85 NR1H2 (1.00) NR1H2NR1H3RXRAPPARGPTGDR2
SCHEMBL4017293 0.83 NR1H2 (0.74) NR1H2NR1H3RXRAPPARGPTGDR2
SCHEMBL4017853 0.83 NR1H2 (0.81) NR1H2NR1H3RXRAPPARGPTGDR2
SCHEMBL4019155 0.83 NR1H2 (0.81) NR1H2NR1H3
SCHEMBL4018567 0.81 NR1H2 (1.00) NR1H2NR1H3RXRAPPARG
SCHEMBL4012201 0.81 NR1H2 (0.84) NR1H2NR1H3RXRAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed