SCHEMBL4014295

SCHEMBL4014295

Nc1ncc(-c2cccc(-c3ccn[nH]3)c2)nc1-c1nc2ccccc2[nH]1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATR Q13535 18/20 0.69
PRKDC P78527 1/20 0.55
ATM Q13315 1/20 0.55
AURKA O14965 1/20 0.52
CDK1 P06493 1/20 0.52
CDK2 P24941 1/20 0.52
AURKB Q96GD4 1/20 0.52
EGFR P00533 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2484717 0.82 ATR (1.00) ATRPRKDCATMCDK1CDK2
SCHEMBL3979058 0.81 ATR (0.76) ATRPRKDCATMCDK1CDK2
SCHEMBL2509897 0.81 ATR (1.00) ATRPRKDCATMCDK1CDK2
SCHEMBL19672786 0.81 ATR (0.71) ATRPRKDCATMCDK1CDK2
SCHEMBL3054972 0.79 ATR (1.00) ATRPRKDCATM
SCHEMBL4006257 0.79 ATR (0.74) ATRPRKDCATMCDK1CDK2
SCHEMBL2681744 0.78 CDK1 (0.70) ATRAURKACDK1CDK2AURKB
SCHEMBL2513033 0.77 ATR (1.00) ATRPRKDCATM
SCHEMBL3469604 0.77 ATR (0.76) ATRPRKDCATMCDK1CDK2
SCHEMBL4436195 0.76 ATR (0.67) ATRPRKDCATMEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO disclosed