SCHEMBL4014748

SCHEMBL4014748

Cc1ccc2c(N3CCC(NC(=O)[C@H]4CCCO4)CC3)nc(-c3ccccc3C(F)F)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.40
ALDH1A1 P00352 10/20 0.40
HPGD P15428 5/20 0.40
GAA P10253 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
ATM Q13315 3/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
RAB9A P51151 4/20 0.39
MAPK1 P28482 3/20 0.39
KMT2A Q03164 1/20 0.39
USP2 O75604 3/20 0.39
HSD17B10 Q99714 3/20 0.39
TP53 P04637 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 3/20 0.38
CYP2C19 P33261 2/20 0.38
TSHR P16473 2/20 0.38
CASP7 P55210 2/20 0.38
CYP1A2 P05177 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13157344 1.00 KDM4E (0.40) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL13769346 1.00 KDM4E (0.40) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL12721405 0.89 SMAD3 (0.46) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL1622793 0.89 SMAD3 (0.46) KDM4EALDH1A1HPGDGAATDP1
Hydrochloric Acid SCHEMBL1623593 0.88 SMAD3 (0.46) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL1622527 0.84 CHEK2 (0.47) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL1623611 0.84 CHEK2 (0.47) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL12723066 0.84 CHEK2 (0.47) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL12723070 0.84 CHEK2 (0.47) KDM4EALDH1A1HPGDGAATDP1
SCHEMBL1623607 0.84 CHEK2 (0.47) KDM4EALDH1A1HPGDGAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed
WO-2006028904-A9 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2006-06-22 WO disclosed