SCHEMBL4015802

SCHEMBL4015802

COc1cc(N2CCN(C(C=O)n3nc(C(F)(F)F)c(Cl)c3C)CC2)ccc1Cl

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.60
CYP2C19 P33261 1/20 0.60
KCNH2 Q12809 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171132 0.92 CCR1 (0.51) CCR1CYP2C19KCNH2
SCHEMBL4020445 0.92 CCR1 (0.60) CCR1CYP2C19KCNH2
SCHEMBL6167744 0.91 CCR1 (0.62) CCR1CYP2C19KCNH2
SCHEMBL4304953 0.91 CCR1 (0.61) CCR1CYP2C19KCNH2
SCHEMBL6193030 0.90 CCR1 (0.62) CCR1CYP2C19KCNH2
SCHEMBL4020420 0.90 CCR1 (0.52) CCR1CYP2C19KCNH2
SCHEMBL4013644 0.89 CCR1 (0.48) CCR1CYP2C19KCNH2
SCHEMBL4022521 0.89 CCR1 (0.62) CCR1CYP2C19KCNH2
SCHEMBL5450338 0.89 CCR1 (0.54) CCR1CYP2C19KCNH2
SCHEMBL4016053 0.88 CCR1 (0.57) CCR1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1691810-A4 SUBSTITUTED PIPERAZINES CHEMOCENTRYX INC (US) 2009-07-01 EP disclosed
EP-1691810-A1 SUBSTITUTED PIPERAZINES ChemoCentryx Inc (US) 2006-08-23 EP disclosed
WO-2005056015-A1 SUBSTITUTED PIPERAZINES CHEMOCENTRYX, INC. (US) 2005-06-23 WO disclosed