SCHEMBL402039

SCHEMBL402039

CCOC(=O)c1cc(Br)c(O)c(C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.55
CA12 O43570 3/20 0.53
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
CA7 P43166 3/20 0.53
CA9 Q16790 3/20 0.53
CA14 Q9ULX7 3/20 0.53
PTPN1 P18031 4/20 0.50
AKR1C4 P17516 2/20 0.50
AKR1C3 P42330 2/20 0.50
AKR1C2 P52895 2/20 0.50
AKR1C1 Q04828 2/20 0.50
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
TTR P02766 1/20 0.46
PTPN2 P17706 2/20 0.46
PTPN11 Q06124 1/20 0.46
ESR2 Q92731 1/20 0.45
TSHR P16473 2/20 0.44
HSD17B10 Q99714 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL401407 0.86 ESR1 (0.54) ESR1CA12CA1CA2CA7
SCHEMBL399551 0.84 CA12 (0.56) ESR1CA12CA1CA2CA7
SCHEMBL16742163 0.82 PTPN11 (0.65) ESR1CA12CA1CA2CA7
SCHEMBL27717216 0.81 CA12 (0.53) ESR1CA12CA1CA2CA7
SCHEMBL27603824 0.80 CA12 (0.58) ESR1CA12CA1CA2CA7
SCHEMBL5990256 0.79 ESR1 (0.58) ESR1CA12CA1CA2CA7
SCHEMBL21487381 0.79 ESR1 (0.56) ESR1CA12CA1CA2CA7
SCHEMBL2821387 0.79 CA12 (0.54) ESR1CA12CA1CA2CA7
SCHEMBL403026 0.77 HSD17B10 (0.42) ESR1CA12CA1CA2CA7
SCHEMBL11763447 0.75 TSHR (0.59) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107935840-B 4-hydroxyisophthalic acid derivative and synthetic method thereof 常州工程职业技术学院 2021-05-25 CN claimed
CN-107935840-B 4-hydroxyisophthalic acid derivative and synthetic method thereof 常州工程职业技术学院 2021-05-25 CN disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
US-20060089392-A1 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089392-A1 Ester derivatives and medicinal use thereof MTTP, CETP, LIPA ESR1 3783/4885CA12 4553/4885CA1 4454/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.