SCHEMBL4020707

SCHEMBL4020707

CC(C)=CCn1c(N2CCCC(N)C2)nc2c1c(=O)n(CC(=O)OCc1ccncc1)c(=O)n2C

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.71
CHRM1 P11229 4/20 0.69
CHRM2 P08172 1/20 0.69
CHRM3 P20309 1/20 0.69
KCNH2 Q12809 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL556113 0.89 DPP4 (0.88) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556105 0.89 DPP4 (0.88) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556791 0.88 DPP4 (0.75) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555632 0.86 DPP4 (0.77) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555212 0.86 DPP4 (0.77) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL556506 0.84 DPP4 (0.82) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555522 0.83 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555869 0.83 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL555920 0.83 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2
SCHEMBL14392635 0.83 DPP4 (0.81) DPP4CHRM1CHRM2CHRM3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7560450-B2 Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO., KG (DE) 2009-07-14 US disclosed
EP-1565468-A1 NOVEL XANTHIN DERIVATIVES, PRODUCTION AND USE THEREOF AS MEDICAMENTS Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2005-08-24 EP disclosed
WO-2004046148-A1 NOVEL XANTHIN DERIVATIVES, PRODUCTION AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-06-03 WO disclosed