SCHEMBL4023786

SCHEMBL4023786

O=C(O)Nc1cccc2cnccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 10/20 0.64
KMT2A Q03164 3/20 0.63
MEN1 O00255 2/20 0.63
MAPK1 P28482 1/20 0.63
HTT P42858 1/20 0.63
BLM P54132 1/20 0.63
MAPT P10636 6/20 0.61
ALDH1A1 P00352 5/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
KDM4E B2RXH2 5/20 0.58
LMNA P02545 1/20 0.57
CHEK1 O14757 1/20 0.56
PIM1 P11309 1/20 0.56
CDK8 P49336 1/20 0.56
GSK3B P49841 1/20 0.56
CDK7 P50613 1/20 0.56
CDK9 P50750 1/20 0.56
LIMK1 P53667 1/20 0.56
ROCK1 Q13464 1/20 0.56
CLK4 Q9HAZ1 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30114438 1.00 TRPV1 (0.64) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL5660097 0.88 TRPV1 (0.71) TRPV1
SCHEMBL30600745 0.87 TRPV1 (0.52) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL6630943 0.85 TRPV1 (0.59) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL2315592 0.85 KDM4E (0.67) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL4023574 0.85 MAPT (0.62) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL30544195 0.85 KDM4E (0.67) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL17737359 0.84 KMT2A (0.76) TRPV1KMT2AMEN1MAPK1HTT
Hydrochloric Acid SCHEMBL2319974 0.84 KDM4E (0.65) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL13151501 0.83 TRPV1 (0.73) TRPV1KMT2AMEN1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478363-B1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LAB (US) 2009-01-14 EP claimed
CN-116096372-A EGFR inhibitor, preparation method and pharmaceutical application thereof 上海和誉生物医药科技有限公司 2023-05-09 CN disclosed
CN-106661018-B Pyrrolo- [2,3-C] pyridine as neurofibrillary tangles imaging agent 默沙东公司 2019-07-19 CN disclosed
CN-106661018-A Pyrrolo[2,3-c]pyridines as imaging agents for neurofibrilary tangles 默沙东公司 2017-05-10 CN disclosed