SCHEMBL4030720

SCHEMBL4030720

CCC(C(=O)NCc1ccc(CN(Cc2ncc(Cl)cc2C)[C@H]2CCCc3cccnc32)c(CO)c1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 18/20 0.44
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2084799 1.00 CXCR4 (0.44) CXCR4MEN1KMT2APOLB
SCHEMBL2084800 1.00 CXCR4 (0.44) CXCR4MEN1KMT2APOLB
SCHEMBL2084796 1.00 CXCR4 (0.44) CXCR4MEN1KMT2APOLB
SCHEMBL2084324 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB
SCHEMBL2084325 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB
SCHEMBL23428716 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB
SCHEMBL2083850 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB
SCHEMBL12935741 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB
SCHEMBL2083848 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB
SCHEMBL2083846 0.94 CXCR4 (0.50) CXCR4MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed