SCHEMBL4031099

SCHEMBL4031099

CNC(=O)c1ccc2cc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 13/20 0.52
CYP3A4 P08684 11/20 0.52
ACSS2 Q9NR19 4/20 0.41
SIRT2 Q8IXJ6 1/20 0.38
PTPN1 P18031 1/20 0.37
PLK1 P53350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312979 0.93 CYP17A1 (0.46) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL4027411 0.91 CYP3A4 (0.53) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL313157 0.91 CYP17A1 (0.45) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL5750054 0.90 CYP3A4 (0.49) CYP17A1CYP3A4SIRT2
SCHEMBL4026360 0.90 CYP3A4 (0.42) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL4033446 0.90 CYP17A1 (0.45) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL4036889 0.90 CYP17A1 (0.45) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL4025229 0.90 CYP3A4 (0.43) CYP17A1CYP3A4ACSS2SIRT2PTPN1
SCHEMBL4024055 0.90 CYP17A1 (0.55) CYP17A1CYP3A4ACSS2SIRT2
SCHEMBL4031717 0.90 CYP3A4 (0.43) CYP17A1CYP3A4ACSS2SIRT2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed