SCHEMBL4033918

SCHEMBL4033918

Cc1nsc2ccc(Nc3ncnc4cccc(OC5CCN(C)CC5)c34)cc12

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.65
ERBB2 P04626 10/20 0.65
KCNH2 Q12809 1/20 0.58
SRC P12931 4/20 0.55
KDR P35968 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5664053 0.99 EGFR (0.64) EGFRERBB2KCNH2SRCKDR
SCHEMBL4037044 0.83 EGFR (0.66) EGFRERBB2KCNH2SRC
Hydrochloric Acid SCHEMBL4034029 0.82 EGFR (0.70) EGFRERBB2KCNH2SRCKDR
SCHEMBL4029893 0.81 ERBB2 (0.70) EGFRERBB2KCNH2SRCKDR
SCHEMBL4039826 0.81 EGFR (0.70) EGFRERBB2KCNH2SRCKDR
SCHEMBL4036837 0.81 EGFR (0.65) EGFRERBB2KCNH2SRCKDR
SCHEMBL4029084 0.80 EGFR (0.70) EGFRERBB2KCNH2SRCKDR
SCHEMBL4032431 0.79 EGFR (0.72) EGFRERBB2KCNH2SRCKDR
Hydrochloric Acid SCHEMBL4037466 0.79 EGFR (0.78) EGFRERBB2KCNH2SRCKDR
Hydrochloric Acid SCHEMBL4041008 0.79 EGFR (0.75) EGFRERBB2KCNH2SRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444211-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-01-21 EP disclosed
EP-1444211-A2 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS AstraZeneca AB (SE) 2004-08-11 EP disclosed
WO-2003040109-A2 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2003-05-15 WO disclosed