SCHEMBL4034166

SCHEMBL4034166

CSCc1cccc(Nc2nccc(N(C)c3ccc4c(C)n[nH]c4c3)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 19/20 0.50
CYP3A4 P08684 3/20 0.50
CYP2D6 P10635 3/20 0.50
CYP2C9 P11712 3/20 0.50
CYP2C19 P33261 3/20 0.50
EPHB4 P54760 1/20 0.49
KIT P10721 7/20 0.48
PDGFRA P16234 7/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12999190 0.89 KDR (0.51) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL31672451 0.87 KDR (0.62) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10151178 0.87 KDR (0.62) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL588358 0.85 KDR (0.55) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL31672434 0.85 KDR (0.54) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10151180 0.85 KDR (0.54) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10187184 0.83 KDR (0.51) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL589306 0.81 KDR (0.53) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL31672519 0.81 KDR (0.51) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6098657 0.81 KDR (0.66) KDRCYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343782-B1 PYRIMIDINEAMINES AS ANGIOGENESIS MODULATORS SMITHKLINE BEECHAM CORP (US) 2009-05-06 EP disclosed