SCHEMBL4035520

SCHEMBL4035520

CN(C)CCCOc1cc(F)c(-c2c(Cl)n[c]nc2NCC(F)(F)F)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.35
CACNA1B Q00975 3/20 0.32
KDM4E B2RXH2 2/20 0.31
EGFR P00533 1/20 0.31
PDK2 Q15119 1/20 0.30
CXCR1 P25024 1/20 0.30
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018949 0.83 KCNH2 (0.35) MAPTCACNA1BKDM4EEGFR
SCHEMBL4016367 0.81 ESR1 (0.35) MAPTCACNA1BKDM4EPDK2
SCHEMBL4020389 0.79 MAPT (0.32) MAPT
Hydrochloric Acid SCHEMBL4025709 0.78 MAPT (0.31) MAPT
Trifluoroacetic Acid SCHEMBL4025752 0.78 CACNA1B (0.39) CACNA1BKDM4EALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL4025706 0.78 MAPT (0.31) MAPT
SCHEMBL4018558 0.77 LIMK1 (0.37) MAPTHRH3
SCHEMBL15626284 0.77 FFAR1 (0.38) CACNA1BALDH1A1
SCHEMBL4017091 0.76 MAPT (0.31) MAPT
SCHEMBL4020578 0.76 CYP1A2 (0.42) CACNA1BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663241-B1 5-ARYLPYRIMIDINES AS ANTICANCER AGENTS WYETH CORP (US) 2009-05-27 EP disclosed