SCHEMBL4036360

SCHEMBL4036360

COc1cc(N2CCOCC2)ccc1Nc1nc(N)n(-c2cccc(C)n2)n1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 6/20 0.67
KIT P10721 5/20 0.67
IRAK4 Q9NWZ3 4/20 0.67
AURKA O14965 1/20 0.67
JAK2 O60674 1/20 0.55
INSR P06213 2/20 0.52
ALK Q9UM73 2/20 0.52
TTK P33981 4/20 0.51
LRRK2 Q5S007 3/20 0.51
PTK2 Q05397 1/20 0.48
DCLK1 O15075 1/20 0.47
MAPK7 Q13164 1/20 0.47
MAPK8 P45983 1/20 0.47
MAPK9 P45984 1/20 0.47
MAPK10 P53779 1/20 0.47
TNK2 Q07912 1/20 0.46
IGF1R P08069 1/20 0.46
ULK1 O75385 1/20 0.46
EGFR P00533 1/20 0.46
ZAP70 P43403 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779714 0.88 FLT3 (0.63) FLT3KITIRAK4AURKAJAK2
SCHEMBL4040811 0.87 FLT3 (0.86) FLT3KITIRAK4AURKAJAK2
SCHEMBL4038234 0.83 FLT3 (0.72) FLT3KITIRAK4AURKAJAK2
SCHEMBL4038723 0.81 FLT3 (0.55) FLT3KITIRAK4AURKAJAK2
SCHEMBL4041811 0.81 FLT3 (0.68) FLT3KITIRAK4AURKAJAK2
SCHEMBL4048022 0.80 FLT3 (1.00) FLT3KITIRAK4AURKAJAK2
SCHEMBL2086723 0.80 FLT3 (1.00) FLT3KITIRAK4AURKAJAK2
SCHEMBL4042645 0.79 FLT3 (0.73) FLT3KITIRAK4AURKAJAK2
SCHEMBL4038386 0.79 FLT3 (0.59) FLT3KITIRAK4AURKAJAK2
SCHEMBL4037633 0.79 FLT3 (0.60) FLT3KITIRAK4AURKAJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed