SCHEMBL4037484

SCHEMBL4037484

COc1cccc(-c2cc(CNc3ncc(Cl)c(Nc4cc(C)[nH]n4)n3)on2)c1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 20/20 0.66
FGFR1 P11362 7/20 0.66
KDR P35968 7/20 0.66
INSR P06213 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2121059 0.89 IGF1R (0.81) IGF1RFGFR1KDRINSR
SCHEMBL4037067 0.86 IGF1R (0.69) IGF1RFGFR1KDRINSR
SCHEMBL2122601 0.84 IGF1R (0.67) IGF1RFGFR1KDRINSR
SCHEMBL2122642 0.82 IGF1R (0.72) IGF1RFGFR1KDRINSR
SCHEMBL3866935 0.81 IGF1R (0.69) IGF1RFGFR1KDRINSR
SCHEMBL2121130 0.80 IGF1R (1.00) IGF1RFGFR1KDRINSR
SCHEMBL4208194 0.79 IGF1R (1.00) IGF1RFGFR1KDRINSR
SCHEMBL4034359 0.79 IGF1R (0.66) IGF1RFGFR1KDRINSR
SCHEMBL4032551 0.77 IGF1R (0.79) IGF1RFGFR1KDRINSR
SCHEMBL2123793 0.77 IGF1R (0.78) IGF1RFGFR1KDRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1456182-B1 PYRIMIDINE DERIVATIVES AS MODULATORS OF INSULINE-LIKE GROWTH FACTOR-1 RECEPTOR (IGF-I) ASTRAZENECA AB (SE) 2009-03-11 EP disclosed