SCHEMBL4040697

SCHEMBL4040697

O=C(NC1CCCCC1)C(C1CCCCC1)C1(c2ccc(F)c(F)c2)Nc2ccccc2N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.44
RAB9A P51151 6/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.42
EPHX2 P34913 3/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
KCNH2 Q12809 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
HTT P42858 2/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HSD17B10 Q99714 1/20 0.38
C3AR1 Q16581 2/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039953 0.90 NPC1 (0.40) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4044713 0.90 KMT2A (0.44) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4044551 0.90 CYP3A4 (0.42) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4044492 0.90 KMT2A (0.42) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4037646 0.89 EPHX2 (0.42) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4037831 0.88 KMT2A (0.42) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL4038973 0.87 NPC1 (0.46) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4037071 0.87 EPHX1 (0.46) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4034552 0.86 NPC1 (0.41) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL4042732 0.86 NR1H4 (0.44) NPC1RAB9ASMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038259-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F.HOFFMANN-LA ROCHE AG (CH) 2009-03-25 EP disclosed
WO-2008000643-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F. HOFFMANN-LA ROCHE AG (CH) 2008-01-03 WO disclosed