SCHEMBL4041224

SCHEMBL4041224

CN1CCC(Oc2cc(N3CC[C@@H](N(C)C)C3)cc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c23)CC1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.73
ERBB2 P04626 9/20 0.73
KCNH2 Q12809 1/20 0.54
GAK O14976 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036765 0.87 EGFR (0.69) EGFRERBB2KCNH2
SCHEMBL4037607 0.86 EGFR (0.84) EGFRERBB2KCNH2GAK
SCHEMBL4038197 0.84 EGFR (0.82) EGFRERBB2KCNH2GAK
SCHEMBL5662192 0.84 EGFR (0.55) EGFRERBB2KCNH2
SCHEMBL4037101 0.84 EGFR (0.81) EGFRERBB2KCNH2GAK
Hydrochloric Acid SCHEMBL5663181 0.83 EGFR (0.55) EGFRERBB2KCNH2
SCHEMBL4031651 0.83 EGFR (0.92) EGFRERBB2KCNH2GAK
SCHEMBL4036105 0.82 EGFR (0.79) EGFRERBB2KCNH2GAK
SCHEMBL4031693 0.82 EGFR (0.79) EGFRERBB2KCNH2GAK
SCHEMBL4034225 0.82 EGFR (0.78) EGFRERBB2KCNH2GAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444211-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-01-21 EP disclosed