SCHEMBL4041316

SCHEMBL4041316

Cc1cccc(-n2nc(Nc3ccccc3Cl)nc2N)n1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 10/20 0.70
IRAK4 Q9NWZ3 6/20 0.70
AURKA O14965 3/20 0.70
KIT P10721 6/20 0.50
TSHR P16473 1/20 0.42
AXL P30530 2/20 0.40
JAK2 O60674 2/20 0.40
BACE1 P56817 2/20 0.39
MAP4K4 O95819 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
GSK3B P49841 1/20 0.39
JAK3 P52333 1/20 0.39
TTK P33981 1/20 0.38
PTK2 Q05397 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4040213 0.82 FLT3 (1.00) FLT3IRAK4AURKAKITAXL
SCHEMBL12779726 0.82 FLT3 (0.65) FLT3IRAK4AURKAKITTSHR
SCHEMBL4038723 0.75 FLT3 (0.55) FLT3IRAK4AURKAKITAXL
SCHEMBL4042028 0.74 FLT3 (0.74) FLT3IRAK4AURKAKITAXL
SCHEMBL4040821 0.73 FLT3 (1.00) FLT3IRAK4AURKAKITTSHR
SCHEMBL4045278 0.72 FLT3 (0.73) FLT3IRAK4AURKAKITTSHR
SCHEMBL12779700 0.72 FLT3 (0.73) FLT3IRAK4AURKAKITTSHR
SCHEMBL4038854 0.71 FLT3 (0.72) FLT3IRAK4AURKAKITAXL
SCHEMBL4040196 0.71 FLT3 (0.48) FLT3IRAK4AURKAKITAXL
SCHEMBL4042908 0.70 MAPT (0.47) FLT3IRAK4AURKAKITTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed