SCHEMBL4042453

SCHEMBL4042453

NCc1cc(-c2ccccc2OC(F)(F)F)no1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.51
SCN9A Q15858 4/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2E1 P05181 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2B6 P20813 1/20 0.43
S1PR1 P21453 3/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CNR2 P34972 1/20 0.41
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
CA12 O43570 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2123714 0.81 NOTUM (0.55) NOTUMCYP2C9CYP2C19CYP2E1CYP2A6
SCHEMBL2120380 0.79 NOTUM (0.53) NOTUMCYP2C9CYP2C19CYP2E1CYP2A6
SCHEMBL4037075 0.78 NOTUM (0.55) NOTUMSCN9ACYP2C9CYP2C19CYP2E1
SCHEMBL16482130 0.78 S1PR1 (0.50) SCN9ACYP2C9CYP2C19S1PR1CYP1A2
SCHEMBL2120898 0.76 NOTUM (0.60) NOTUMCYP2C9CYP2C19CYP2E1CYP2A6
SCHEMBL30093453 0.76 S1PR1 (0.45) SCN9ACYP2C9CYP2C19S1PR1CYP1A2
SCHEMBL28214769 0.75 HCRTR1 (0.48) SCN9ACYP2C9S1PR1CYP3A4CYP2D6
SCHEMBL4036299 0.75 NTRK1 (0.40) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL27612624 0.74 NOTUM (0.62) NOTUMCYP2C9CYP2C19CYP2E1CYP2A6
SCHEMBL1221395 0.74 NPC1 (0.36) SCN9ACYP2C9CYP2C19S1PR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1456182-B1 PYRIMIDINE DERIVATIVES AS MODULATORS OF INSULINE-LIKE GROWTH FACTOR-1 RECEPTOR (IGF-I) ASTRAZENECA AB (SE) 2009-03-11 EP disclosed