Bicarbonate

Bicarbonate

SCHEMBL4044942

O=C(O)O.O=C1CSc2ccc(CN[C@H]3CCCC[C@H]3O)nc2N1

nearest known ligand 0.46

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.41
TRPV3 Q8NET8 7/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL4045725 1.00 KCNH2 (0.41) KCNH2TRPV3
Bicarbonate SCHEMBL4043287 1.00 KCNH2 (0.41) KCNH2TRPV3
SCHEMBL5264047 0.85 KCNH2 (0.38) KCNH2
SCHEMBL3579608 0.85 KCNH2 (0.38) KCNH2
SCHEMBL3581981 0.85 KCNH2 (0.38) KCNH2
SCHEMBL3573905 0.85 KCNH2 (0.38) KCNH2
Bicarbonate SCHEMBL5738279 0.81 KCNH2 (0.40) KCNH2
Bicarbonate SCHEMBL5738348 0.81 KCNH2 (0.40) KCNH2
SCHEMBL5262915 0.81 KCNH2 (0.38) KCNH2TRPV3
SCHEMBL5259010 0.81 KCNH2 (0.38) KCNH2TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463728-B1 FUSED CYCLIC MODULATORS OF NUCLEAR HORMONE RECEPTOR FUNCTION BRISTOL MYERS SQUIBB CO (US) 2009-01-14 EP disclosed