SCHEMBL4045741

SCHEMBL4045741

Nc1nc(-c2ccco2)c2nnn(Cc3cc(CNC(=O)O)ccn3)c2n1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.66
ADORA2B P29275 20/20 0.66
ADORA1 P30542 20/20 0.66
ADORA3 P0DMS8 19/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047878 0.89 ADORA2A (0.75) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4045607 0.88 ADORA2A (0.76) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4048192 0.88 ADORA2A (0.59) ADORA2AADORA2BADORA1ADORA3
SCHEMBL14143125 0.85 ADORA2A (0.79) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4045860 0.84 ADORA2A (0.72) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4045360 0.83 ADORA2A (0.73) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4047636 0.83 ADORA2A (0.76) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4053505 0.82 ADORA2A (0.61) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4044825 0.81 ADORA2A (0.72) ADORA2AADORA2BADORA1ADORA3
SCHEMBL4047232 0.81 ADORA2A (0.76) ADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-B1 TRIAZOLO 4,5-d PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2009-03-04 EP claimed