SCHEMBL4045757

SCHEMBL4045757

Nc1nc(-c2cc[nH]n2)c2nnn(Cc3cccc([N+](=O)[O-])c3)c2n1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.67
ADORA1 P30542 19/20 0.67
ADORA3 P0DMS8 17/20 0.67
ADORA2B P29275 17/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4045738 0.99 ADORA2A (0.66) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4050324 0.85 ADORA2A (0.63) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4045835 0.84 ADORA2A (0.53) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4052225 0.84 ADORA2A (0.68) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL2990319 0.84 ADORA2A (0.73) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4457050 0.83 ADORA2A (0.67) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL13707441 0.81 ADORA2A (0.67) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4052560 0.81 ADORA2A (0.69) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL2984371 0.81 ADORA2A (0.66) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL2983643 0.80 ADORA2A (0.68) ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-B1 TRIAZOLO 4,5-d PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2009-03-04 EP claimed